34562-97-5

  • Product Name:Pikamilone
  • Molecular Formula:C10H12N2O3
  • Purity:99%
  • Molecular Weight:208.217
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Product Details

Melting Point:210-212oC

Appearance:white crystalline powder

Purity:99%

Buy Quality Pikamilone 34562-97-5 In Stock with Immediately Delivery

  • Molecular Formula:C10H12N2O3
  • Molecular Weight:208.217
  • Appearance/Colour:white crystalline powder 
  • Vapor Pressure:9.65E-12mmHg at 25°C 
  • Melting Point:210-212oC 
  • Boiling Point:522.4 °C at 760 mmHg 
  • PKA:4.60±0.10(Predicted) 
  • Flash Point:269.8 °C 
  • PSA:79.29000 
  • Density:1.245 g/cm3 
  • LogP:1.06710 

Pikamilone(Cas 34562-97-5) Usage

InChI:InChI=1/C10H12N2O3.Na/c13-9(14)4-2-6-12-10(15)8-3-1-5-11-7-8;/h1,3,5,7H,2,4,6H2,(H,12,15)(H,13,14);/q;+1/p-1

34562-97-5 Relevant articles

Evaluation of isonicotinoyl-γ-aminobutyric acid (GABA) nicotinoyl-GABA as pro-drugs of GABA

Matsuyama,Yamashita,Noda,Goto,Ichimaru,Gomita

, p. 4089 - 4095 (1984)

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Synthesis and biological evaluation of GABA derivatives able to cross the blood-Brain barrier in rats

Carelli, Vincenzo,Liberatore, Felice,Scipione, Luigi,Giorgioni, Gianfabio,Di Stefano, Antonio,Impicciatore, Mariannina,Ballabeni, Vigilio,Calcina, Francesco,Magnanini, Francesca,Barocelli, Elisabetta

, p. 3765 - 3769 (2003)

Two new GABA derivatives, 1 and 2, were ...

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Page/Page column 52; 53, (2011/08/08)

Novel small molecule compounds for reduc...

34562-97-5 Process route

nicotinoyl chloride
121667-28-5

nicotinoyl chloride

N-nicotinoyl-gamma-aminobutyric acid
34562-97-5

N-nicotinoyl-gamma-aminobutyric acid

Conditions
Conditions Yield
With palladium 10% on activated carbon; hydrogen; In methanol; at 20 ℃; for 2h; Inert atmosphere;
90%
With palladium 10% on activated carbon; hydrogen; In methanol; at 20 ℃; for 2h;
90%
With hydrogen; palladium on activated charcoal;
4-[(pyridine-3-carbonyl)amino]butyric acid methyl ester

4-[(pyridine-3-carbonyl)amino]butyric acid methyl ester

N-nicotinoyl-gamma-aminobutyric acid
34562-97-5

N-nicotinoyl-gamma-aminobutyric acid

Conditions
Conditions Yield
4-[(pyridine-3-carbonyl)amino]butyric acid methyl ester; With water; lithium hydroxide; In tetrahydrofuran; at 25 - 45 ℃;
With hydrogenchloride; In water; pH=2 - 3;
80%

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